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概述选择性和非选择性CNS-Pharmacodynamic概要的GABA受体激动剂
表4
眼跳峰值速度变化的结果线性模型从基线和日志的身体摇摆变化从基线治疗治疗由SPV变化从基线交互。
|
| 治疗 |
ΔSPV-relative关系 |
项 |
估计的治疗 |
氯羟去甲安定的估计 |
价值 |
|
| TPA023 1.5毫克 |
ΔSway-ΔSPV |
坡 |
−0.00048 |
−0.00305 |
< 0.0001 |
| 拦截 |
−0.01316 |
0.1292 |
< 0.0001 |
| ΔVAS警觉性-ΔSPV |
坡 |
0.03312 |
0.126 |
0.0001 |
| 拦截 |
0.4551 |
−4.4739 |
0.0021 |
|
| TPACMP2 0.75毫克 |
ΔSway-ΔSPV |
坡 |
−0.00027 |
−0.00305 |
< 0.0001 |
| 拦截 |
0.03784 |
0.1292 |
0.0009 |
| ΔVAS警觉性-ΔSPV |
坡 |
0.09884 |
0.126 |
0.2525 |
| 拦截 |
−1.4465 |
−4.4739 |
0.0397 |
|
| SL65.1498 25毫克 |
ΔSway-ΔSPV |
坡 |
−0.00128 |
−0.00305 |
0.0003 |
| 拦截 |
0.0222 |
0.1292 |
< 0.0001 |
| ΔVAS警觉性-ΔSPV |
坡 |
0.04193 |
0.126 |
0.0009 |
| 拦截 |
0.2453 |
−4.4739 |
< 0.0001 |
| ΔSmooth-ΔSPV |
坡 |
0.01554 |
0.1099 |
< 0.0001 |
| 拦截 |
−1.4483 |
−6.2553 |
< 0.0001 |
|
| 阿普唑仑1毫克 |
ΔSway-ΔSPV |
坡 |
−0.00204 |
−0.00305 |
0.0667 |
| 拦截 |
0.001788 |
0.1292 |
< 0.0001 |
| ΔVAS警觉性-ΔSPV |
坡 |
0.0734 |
0.126 |
0.0763 |
| 拦截 |
−0.628 |
−4.4739 |
0.0254 |
| ΔTrack-ΔSPV |
坡 |
0.0747 |
0.0572 |
0.1545 |
| 拦截 |
0.3023 |
−4.0742 |
< 0.0001 |
| ΔSmooth-ΔSPV |
坡 |
0.08077 |
0.1099 |
0.2808 |
| 拦截 |
−1.4025 |
−6.2553 |
0.0002 |
|
| 唑吡坦10毫克 |
ΔSway-ΔSPV |
坡 |
−0.0033 |
−0.00305 |
0.7336 |
| 拦截 |
0.06014 |
0.1292 |
0.0127 |
| ΔVAS警觉性-ΔSPV |
坡 |
0.1526 |
0.126 |
0.5231 |
| 拦截 |
−3.2697 |
−4.4739 |
0.5219 |
| ΔTrack-ΔSPV |
坡 |
0.0489 |
0.0572 |
0.6240 |
| 拦截 |
−0.9123 |
−4.0742 |
< 0.0001 |
| ΔSmooth-ΔSPV |
坡 |
0.09771 |
0.1099 |
0.7412 |
| 拦截 |
−3.8439 |
−6.2553 |
0.0815 |
|
|